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Janez Ilaš
Janez Ilaš
Professor of Medicinal Chemistry, Faculty of Pharmacy, University of Ljubljana
Verified email at ffa.uni-lj.si
Title
Cited by
Cited by
Year
Recent advances in the synthesis of 2H-1, 4-benzoxazin-3-(4H)-ones and 3, 4-dihydro-2H-1, 4-benzoxazines
J Ilaš, PŠ Anderluh, MS Dolenc, D Kikelj
Tetrahedron 61 (31), 7325-7348, 2005
1962005
Dual inhibitors of human DNA topoisomerase II and other cancer-related targets
Z Skok, N Zidar, D Kikelj, J Ilaš
Journal of medicinal chemistry 63 (3), 884-904, 2019
1682019
Discovery of benzothiazole scaffold-based DNA gyrase B inhibitors
M Gjorgjieva, T Tomasic, M Barancokova, S Katsamakas, J Ilas, ...
Journal of medicinal chemistry 59 (19), 8941-8954, 2016
1282016
Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site
T Tomasic, S Katsamakas, Z Hodnik, J Ilaš, M Brvar, T Solmajer, ...
Journal of medicinal chemistry 58 (14), 5501-5521, 2015
1252015
A road map for prioritizing warheads for cysteine targeting covalent inhibitors
P Abranyi-Balogh, L Petri, T Imre, P Szijj, A Scarpino, M Hrast, A Mitrović, ...
European journal of medicinal chemistry 160, 94-107, 2018
1172018
Toward a Novel Class of Antithrombotic Compounds with Dual Function. Discovery of 1,4-Benzoxazin-3(4H)-one Derivatives Possessing Thrombin Inhibitory and†…
P Štefanič Anderluh, M Anderluh, J Ilaš, J Mravljak, M Sollner Dolenc, ...
Journal of medicinal chemistry 48 (9), 3110-3113, 2005
802005
Antimicrobial activity of the marine alkaloids, clathrodin and oroidin, and their synthetic analogues
N Zidar, S Montalv„o, Ž Hodnik, DA Nawrot, A Žula, J Ilaš, D Kikelj, ...
Marine drugs 12 (2), 940-963, 2014
702014
3,4-Dihydro-2H-1,4-benzoxazine Derivatives Combining Thrombin Inhibitory and Glycoprotein IIb/IIIa Receptor Antagonistic Activity as a Novel Class of†…
J Ilaš, Z Jakopin, T Borštnar, M Stegnar, D Kikelj
Journal of medicinal chemistry 51 (18), 5617-5629, 2008
692008
N-Phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATP Competitive DNA Gyrase B Inhibitors: Design, Synthesis, and Evaluation
N Zidar, H Macut, T Tomasic, M Brvar, S Montalvao, P Tammela, ...
Journal of medicinal chemistry 58 (15), 6179-6194, 2015
652015
Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors
Ž Jakopin, J Ilaš, M BarančokovŠ, M Brvar, P Tammela, MS Dolenc, ...
European Journal of Medicinal Chemistry 130, 171-184, 2017
642017
Influence of different classes of crosslinkers on alginate polyelectrolyte nanoparticle formation, thermodynamics and characteristics
J Mirtič, J Ilaš, J Kristl
Carbohydrate polymers 181, 93-102, 2018
602018
Synthesis and Evaluation of N‐Phenylpyrrolamides as DNA Gyrase B Inhibitors
M Durcik, P Tammela, M BarančokovŠ, T Tomašič, J Ilaš, D Kikelj, N Zidar
ChemMedChem 13 (2), 186-198, 2018
562018
ATP-competitive DNA gyrase and topoisomerase IV inhibitors as antibacterial agents
M Durcik, T Tomašič, N Zidar, A Zega, D Kikelj, LP Mašič, J Ilaš
Expert opinion on therapeutic patents 29 (3), 171-180, 2019
552019
Recent progress in the discovery and development of DNA gyrase B inhibitors
M BarančokovŠ, D Kikelj, J Ilaš
Future medicinal chemistry 10 (10), 1207-1227, 2018
522018
New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity
M Durcik, D Lovison, Ž Skok, CD Cruz, P Tammela, T Tomašič, DB Tiz, ...
European journal of medicinal chemistry 154, 117-132, 2018
492018
Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitors
T Tomašič, M Mirt, M BarančokovŠ, J Ilaš, N Zidar, P Tammela, D Kikelj
Bioorganic & medicinal chemistry 25 (1), 338-349, 2017
492017
Structure-activity relationships and molecular docking studies of chromene and chromene based azo chromophores: A novel series of potent antimicrobial and anticancer agents
TH Afifi, RM Okasha, HEA Ahmed, J Ilaš, T Saleh, AS Abd-El-Aziz
EXCLI journal 16, 868, 2017
482017
Exploring protein hotspots by optimized fragment pharmacophores
D Bajusz, WS Wade, G Satała, AJ Bojarski, J Ilaš, J Ebner, F Grebien, ...
Nature Communications 12 (1), 3201, 2021
412021
An optimised series of substituted N-phenylpyrrolamides as DNA gyrase B inhibitors
DB Tiz, Ž Skok, M Durcik, T Tomašič, LP Mašič, J Ilaš, A Zega, ...
European journal of medicinal chemistry 167, 269-290, 2019
402019
New N-phenyl-4, 5-dibromopyrrolamides and N-Phenylindolamides as ATPase inhibitors of DNA gyrase
N Zidar, T Tomašič, H Macut, A Sirc, M Brvar, S Montalvao, P Tammela, ...
European Journal of Medicinal Chemistry 117, 197-211, 2016
382016
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