András Váradi
András Váradi
E-mail megerősítve itt: cumc.columbia.edu
Cím
Hivatkozott rá
Hivatkozott rá
Év
Mitragynine/corynantheidine pseudoindoxyls as opioid analgesics with mu agonism and delta antagonism, which do not recruit β-arrestin-2
A Váradi, GF Marrone, TC Palmer, A Narayan, MR Szabó, V Le Rouzic, ...
Journal of medicinal chemistry 59 (18), 8381-8397, 2016
1072016
Synthetic and Receptor Signaling Explorations of the Mitragyna Alkaloids: Mitragynine as an Atypical Molecular Framework for Opioid Receptor Modulators
AC Kruegel, MM Gassaway, A Kapoor, A Váradi, S Majumdar, M Filizola, ...
Journal of the American Chemical Society 138 (21), 6754-6764, 2016
1032016
Detection and identification of the new potential synthetic cannabinoids 1-pentyl-3-(2-iodobenzoyl) indole and 1-pentyl-3-(1-adamantoyl) indole in seized bulk powders in Hungary
P Jankovics, A Váradi, L Tölgyesi, S Lohner, J Németh-Palotás, J Balla
Forensic science international 214 (1-3), 27-32, 2012
942012
Isocyanide-based multicomponent reactions for the synthesis of heterocycles
A Váradi, TC Palmer, R Notis Dardashti, S Majumdar
Molecules 21 (1), 19, 2016
882016
Identification and characterization of the new designer drug 4′-methylethcathinone (4-MEC) and elaboration of a novel liquid chromatography–tandem mass spectrometry (LC–MS/MS …
P Jankovics, A Váradi, L Tölgyesi, S Lohner, J Németh-Palotás, ...
Forensic Science International 210 (1-3), 213-220, 2011
822011
Three-component coupling approach for the synthesis of diverse heterocycles utilizing reactive nitrilium trapping
A Varadi, TC Palmer, PR Notis, GN Redel-Traub, D Afonin, JJ Subrath, ...
Organic letters 16 (6), 1668-1671, 2014
282014
Synthesis and characterization of a dual kappa-delta opioid receptor agonist analgesic blocking cocaine reward behavior
A Váradi, GF Marrone, SO Eans, ML Ganno, JJ Subrath, V Le Rouzic, ...
ACS chemical neuroscience 6 (11), 1813-1824, 2015
222015
Synthesis of carfentanil amide opioids using the ugi multicomponent reaction
A Váradi, TC Palmer, N Haselton, D Afonin, JJ Subrath, V Le Rouzic, ...
ACS chemical neuroscience 6 (9), 1570-1577, 2015
182015
A novel µ-opioid receptor ligand with high in vitro and in vivo agonist efficacy
E Lacko, A Varadi, R Rapavi, F Zador, P Riba, S Benyhe, A Borsodi, ...
Current medicinal chemistry 19 (27), 4699-4707, 2012
182012
Synthesis and configurational assignment of 1, 2-dihydroimidazo [5, 1-b] quinazoline-3, 9-diones: novel NMDA receptor antagonists
A Váradi, P Horváth, T Kurtán, A Mándi, G Tóth, A Gergely, J Kökösi
Tetrahedron 68 (50), 10365-10371, 2012
172012
Sulfate esters of morphine derivatives: Synthesis and characterization
A Váradi, A Gergely, S Béni, P Jankovics, B Noszál, S Hosztafi
European journal of pharmaceutical sciences 42 (1-2), 65-72, 2011
172011
Mild, Pd-catalyzed stannylation of radioiodination targets
JE Pickett, A Váradi, TC Palmer, SG Grinnell, JM Schrock, GW Pasternak, ...
Bioorganic & medicinal chemistry letters 25 (8), 1761-1764, 2015
142015
Novel 6β-acylaminomorphinans with analgesic activity
A Váradi, S Hosztafi, V Le Rouzic, G Tóth, Á Urai, B Noszál, ...
European journal of medicinal chemistry 69, 786-789, 2013
142013
New morphine analogs produce peripheral antinociception within a certain dose range of their systemic administration
E Lackó, P Riba, Z Giricz, A Váradi, L Cornic, M Balogh, K Király, K Csekő, ...
Journal of Pharmacology and Experimental Therapeutics 359 (1), 171-181, 2016
132016
Genetic dissociation of morphine analgesia from hyperalgesia in mice
GF Marrone, V Le Rouzic, A Varadi, J Xu, AM Rajadhyaksha, S Majumdar, ...
Psychopharmacology 234 (12), 1891-1900, 2017
92017
A non-retinoid antagonist of retinol-binding protein 4 rescues phenotype in a model of Stargardt disease without inhibiting the visual cycle
B Racz, A Varadi, J Kong, R Allikmets, PG Pearson, G Johnson, CL Cioffi, ...
Journal of Biological Chemistry 293 (29), 11574-11588, 2018
82018
New opioid receptor antagonist: Naltrexone-14-O-sulfate synthesis and pharmacology
F Zádor, K Király, A Váradi, M Balogh, Á Fehér, D Kocsis, AI Erdei, ...
European journal of pharmacology 809, 111-121, 2017
62017
Glucosides of morphine derivatives: synthesis and characterization
A Váradi, D Lévai, G Tóth, P Horváth, B Noszál, S Hosztafi
Monatshefte für Chemie-Chemical Monthly 144 (2), 255-262, 2013
42013
14-O-Methylmorphine: a novel selective mu-opioid receptor agonist with high efficacy and affinity
F Zádor, M Balogh, A Váradi, ZS Zádori, K Király, E Szűcs, B Varga, ...
European Journal of Pharmacology 814, 264-273, 2017
32017
Synthesis and pharmacological evaluation of novel selective MOR agonist 6β-pyridinyl amidomorphines exhibiting long-lasting antinociception
Á Urai, A Váradi, L Szőcs, B Komjáti, V Le Rouzic, A Hunkele, ...
MedChemComm 8 (1), 152-157, 2017
32017
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Cikkek 1–20