Screening and biological effects of marine pyrroloiminoquinone alkaloids: Potential inhibitors of the HIF-1α/p300 interaction AKL Goey, CH Chau, TM Sissung, KM Cook, DJ Venzon, A Castro, ... Journal of natural products 79 (5), 1267-1275, 2016 | 59 | 2016 |
Efficacy of a series of alpha-pyrone derivatives against Leishmania (L.) infantum and Trypanosoma cruzi AG Tempone, DD Ferreira, ML Lima, TAC Silva, SET Borborema, ... European Journal of Medicinal Chemistry 139, 947-960, 2017 | 36 | 2017 |
6-Bromoindolglyoxylamido derivatives as antimicrobial agents and antibiotic enhancers SA Li, MM Cadelis, K Sue, M Blanchet, N Vidal, JM Brunel, ... Bioorganic & Medicinal Chemistry 27 (10), 2090-2099, 2019 | 26 | 2019 |
Spermine Derivatives of Indole‐3‐carboxylic Acid, Indole‐3‐acetic Acid and Indole‐3‐acrylic Acid as Gram‐Negative Antibiotic Adjuvants MM Cadelis, SA Li, ML Bourguet‐Kondracki, M Blanchet, H Douafer, ... ChemMedChem 16 (3), 513-523, 2021 | 24 | 2021 |
Preclinical evaluation of discorhabdins in antiangiogenic and antitumor models EM Harris, JD Strope, SL Beedie, PA Huang, AKL Goey, KM Cook, ... Marine Drugs 16 (7), 241, 2018 | 23 | 2018 |
Exploration of the antibiotic potentiating activity of indolglyoxylpolyamines MM Cadelis, EIW Pike, W Kang, Z Wu, ML Bourguet-Kondracki, ... European Journal of Medicinal Chemistry 183, 111708, 2019 | 18 | 2019 |
Epipyrone A, a Broad-Spectrum Antifungal Compound Produced by Epicoccum nigrum ICMP 19927 AJ Lee, MM Cadelis, SH Kim, S Swift, BR Copp, SG Villas-Boas Molecules 25 (24), 5997, 2020 | 16 | 2020 |
Exploration of the electrophilic reactivity of the cytotoxic marine alkaloid discorhabdin C and subsequent discovery of a new dimeric C-1/N-13-linked discorhabdin natural product CFC Lam, MM Cadelis, BR Copp Marine drugs 18 (8), 404, 2020 | 16 | 2020 |
A revised structure and assigned absolute configuration of theissenolactone A MM Cadelis, S Geese, L Gris, BS Weir, BR Copp, S Wiles Molecules 25 (20), 4823, 2020 | 13 | 2020 |
Exploration of the influence of spiro-dienone moiety on biological activity of the cytotoxic marine alkaloid discorhabdin P CFC Lam, MM Cadelis, BR Copp Tetrahedron 73 (32), 4779-4785, 2017 | 13 | 2017 |
Discovery and preliminary structure–activity relationship studies on tecomaquinone I and tectol as novel farnesyltransferase and plasmodial inhibitors MM Cadelis, ML Bourguet-Kondracki, J Dubois, A Valentin, D Barker, ... Bioorganic & Medicinal Chemistry 24 (14), 3102-3107, 2016 | 11 | 2016 |
Repurposing primaquine as a polyamine conjugate to become an antibiotic adjuvant AN Pearce, D Chen, LR Edmeades, MM Cadelis, A Troudi, JM Brunel, ... Bioorganic & Medicinal Chemistry 38, 116110, 2021 | 10 | 2021 |
Antimicrobial Metabolites against Methicillin-Resistant Staphylococcus aureus from the Endophytic Fungus Neofusicoccum australe MM Cadelis, S Geese, BB Uy, DR Mulholland, SJ van de Pas, A Grey, ... Molecules 26 (4), 1094, 2021 | 10 | 2021 |
A review of fungal protoilludane sesquiterpenoid natural products MM Cadelis, BR Copp, S Wiles Antibiotics 9 (12), 928, 2020 | 10 | 2020 |
Structure-activity relationship studies on thiaplidiaquinones A and B as novel inhibitors of Plasmodium falciparum and farnesyltransferase MM Cadelis, ML Bourguet-Kondracki, J Dubois, M Kaiser, JM Brunel, ... Bioorganic & medicinal chemistry 25 (16), 4433-4443, 2017 | 9 | 2017 |
Synthesis of hemitectol, tectol, and tecomaquinone i MM Cadelis, D Barker, BR Copp Synlett 23 (20), 2939-2942, 2012 | 9 | 2012 |
Isolation of a Novel Polyketide from Neodidymelliopsis sp. MM Cadelis, H Gordon, A Grey, S Geese, DR Mulholland, BS Weir, ... Molecules 26 (11), 3235, 2021 | 8 | 2021 |
Synthesis and antibacterial analysis of analogues of the marine alkaloid pseudoceratidine D Barker, S Lee, KG Varnava, K Sparrow, M van Rensburg, RC Deed, ... Molecules 25 (11), 2713, 2020 | 7 | 2020 |
α, ω-Diacyl-Substituted Analogues of Natural and Unnatural Polyamines: Identification of Potent Bactericides That Selectively Target Bacterial Membranes D Chen, MM Cadelis, F Rouvier, T Troia, LR Edmeades, K Fraser, ES Gill, ... International Journal of Molecular Sciences 24 (6), 5882, 2023 | 6 | 2023 |
Valorisation of the diterpene podocarpic acid–Antibiotic and antibiotic enhancing activities of polyamine conjugates SA Li, MM Cadelis, RC Deed, H Douafer, ML Bourguet-Kondracki, ... Bioorganic & Medicinal Chemistry 64, 116762, 2022 | 6 | 2022 |